SCHEMBL7479569

SCHEMBL7479569

Nc1cc(-c2ccc(F)cc2)cc2nc(-c3ccco3)nn12

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.55
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7485299 0.88 ADORA2A (0.56) ADORA2A
SCHEMBL7428821 0.88 ADORA2A (0.55) ADORA2AMAPTKMT2A
SCHEMBL7708822 0.87 ADORA2A (0.52) ADORA2A
SCHEMBL7430360 0.86 ADORA2A (0.56) ADORA2A
SCHEMBL7486297 0.85 ADORA2A (0.52) ADORA2A
SCHEMBL7478123 0.85 ADORA2A (0.52) ADORA2A
SCHEMBL7705895 0.85 ADORA2A (0.52) ADORA2A
SCHEMBL7709135 0.85 ADORA2A (0.58) ADORA2AKMT2A
SCHEMBL7709137 0.84 ADORA2A (0.54) ADORA2A
SCHEMBL7705914 0.84 ADORA2A (0.53) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP claimed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US claimed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO claimed
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed