SCHEMBL7479653

SCHEMBL7479653

CN(C)C(=O)CCN1CCc2ccc(N3CCN([C@H]4CC[C@H](CCC(=O)O)CC4)C3=O)cc2CC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.37
F2 P00734 2/20 0.36
F10 P00742 2/20 0.36
DRD3 P35462 4/20 0.33
ACHE P22303 4/20 0.33
HTR2A P28223 2/20 0.33
PRSS1 P07477 1/20 0.33
HTR1A P08908 1/20 0.33
KCNH2 Q12809 1/20 0.33
DRD4 P21917 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7470901 0.91 F10 (0.39) DRD2F2F10DRD3ACHE
SCHEMBL8564530 0.89 F2 (0.38) DRD2F2F10DRD3ACHE
SCHEMBL8564532 0.89 F2 (0.38) DRD2F2F10DRD3ACHE
SCHEMBL8562349 0.88 F2 (0.39) F2F10ACHE
SCHEMBL8562341 0.88 F2 (0.39) F2F10ACHE
Hydrochloric Acid SCHEMBL8562318 0.88 F10 (0.38) DRD2F2F10DRD3ACHE
SCHEMBL8562653 0.87 F10 (0.39) DRD2F2F10ACHEPRSS1
SCHEMBL8562646 0.87 F10 (0.39) DRD2F2F10ACHEPRSS1
Hydrochloric Acid SCHEMBL8560749 0.87 F2 (0.38) F2F10ACHEPRSS1
Hydrochloric Acid SCHEMBL8560802 0.87 F10 (0.38) DRD2F2F10ACHEPRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed