SCHEMBL7485443

SCHEMBL7485443

COC(=O)c1ccc(CCc2nc(-c3ccccc3)oc2C)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.56
KDM4E B2RXH2 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
PPARG P37231 17/20 0.55
PPARA Q07869 14/20 0.55
PPARD Q03181 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1123237 0.86 PPARG (0.73) PPARGPPARAPPARD
SCHEMBL12469332 0.83 MEN1 (0.54) FFAR1KDM4EMEN1KMT2APPARG
SCHEMBL3278854 0.82 MAPT (0.68) FFAR1PPARGPPARA
SCHEMBL4036791 0.81 PPARG (0.67) PPARGPPARA
SCHEMBL31180905 0.81 MAPT (0.53) FFAR1KDM4EMEN1KMT2APPARG
SCHEMBL6387594 0.81 PPARG (0.69) PPARGPPARAPPARD
SCHEMBL4031706 0.81 KDR (0.57) FFAR1KDM4EPPARGPPARAPPARD
SCHEMBL12469625 0.81 MEN1 (0.54) KDM4EMEN1KMT2APPARGPPARA
SCHEMBL7486859 0.80 KDM4E (0.57) FFAR1KDM4EPPARGPPARAPPARD
SCHEMBL15325997 0.80 MEN1 (0.58) KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP disclosed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed