SCHEMBL7486409

SCHEMBL7486409

COc1ccccc1NC(=S)Nc1ccc(Oc2ccnc3cc(OC)c(OC)cc23)cc1

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 16/20 0.79
KDR P35968 8/20 0.78
KIT P10721 6/20 0.69
MET P08581 1/20 0.66
FGFR2 P21802 3/20 0.64
AXL P30530 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479716 0.92 PDGFRA (0.79) PDGFRAKDRKITMETFGFR2
SCHEMBL7479420 0.91 PDGFRA (0.79) PDGFRAKDRKITMETFGFR2
SCHEMBL7489927 0.88 PDGFRA (1.00) PDGFRAKDRKITMETFGFR2
SCHEMBL7489114 0.88 PDGFRA (1.00) PDGFRAKDR
SCHEMBL1881332 0.86 PDGFRA (0.92) PDGFRAKDRKITAXL
SCHEMBL1876747 0.86 PDGFRA (0.81) PDGFRAKDRKITMETAXL
SCHEMBL7481612 0.84 PDGFRA (0.81) PDGFRAKDRKITMETFGFR2
SCHEMBL2748182 0.84 KDR (0.67) PDGFRAKDRKITMETFGFR2
SCHEMBL5824535 0.83 PDGFRA (0.76) PDGFRAKDRKITMETFGFR2
SCHEMBL5825323 0.83 PDGFRA (0.85) PDGFRAKDRKITMETAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed