SCHEMBL7487347

SCHEMBL7487347

COc1cc2nccc(Oc3ccc(NC(=O)Nc4ccccc4F)cc3)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 19/20 1.00
KDR P35968 18/20 1.00
MET P08581 1/20 0.77
HDAC1 Q13547 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1876335 0.96 PDGFRA (0.93) PDGFRAKDRMETHDAC1
SCHEMBL7479951 0.92 PDGFRA (1.00) PDGFRAKDR
SCHEMBL7489114 0.91 PDGFRA (1.00) PDGFRAKDR
SCHEMBL7489063 0.90 PDGFRA (0.83) PDGFRAKDR
SCHEMBL7483562 0.89 KDR (1.00) PDGFRAKDR
SCHEMBL7477668 0.89 PDGFRA (1.00) PDGFRAKDR
SCHEMBL7481767 0.89 PDGFRA (0.82) PDGFRAKDR
SCHEMBL7483440 0.89 PDGFRA (0.85) PDGFRAKDR
SCHEMBL7480087 0.89 KDR (1.00) PDGFRAKDR
SCHEMBL7485134 0.89 PDGFRA (1.00) PDGFRAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP claimed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US claimed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed