SCHEMBL7487407

SCHEMBL7487407

COc1cc2nccc(Oc3ccc(NC(=O)NCCCCl)cc3)c2cc1OC

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 18/20 0.74
KDR P35968 17/20 0.74
AXL P30530 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3936662 0.92 KDR (0.74) PDGFRAKDR
SCHEMBL5091900 0.91 PDGFRA (0.72) PDGFRAKDRAXL
SCHEMBL4475483 0.91 PDGFRA (0.72) PDGFRAKDR
SCHEMBL7488292 0.90 PDGFRA (0.71) PDGFRAKDR
SCHEMBL6227724 0.90 PDGFRA (0.71) PDGFRAKDR
SCHEMBL6227624 0.90 PDGFRA (0.77) PDGFRAKDR
SCHEMBL1878994 0.90 PDGFRA (0.77) PDGFRAKDRAXL
SCHEMBL4465899 0.89 PDGFRA (0.70) PDGFRAKDR
SCHEMBL5092913 0.89 PDGFRA (0.70) PDGFRAKDR
SCHEMBL7476738 0.89 PDGFRA (0.75) PDGFRAKDRAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed