SCHEMBL748770

SCHEMBL748770

COC(=O)NCC(C)CC(=O)N1CCCC1c1ncc(-c2ccc(Br)cc2)[nH]1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.59
CYP2C9 P11712 3/20 0.59
KCNH2 Q12809 2/20 0.59
NR1I2 O75469 2/20 0.59
ABCB11 O95342 1/20 0.59
OPRK1 P41145 1/20 0.59
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 1/20 0.53
PRCP P42785 11/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL751463 0.89 CYP3A4 (0.49) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL751612 0.89 CYP3A4 (0.56) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL750166 0.88 CYP3A4 (0.57) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL749500 0.88 CYP3A4 (0.79) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL749345 0.88 CYP3A4 (0.44) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL19339668 0.88 CYP3A4 (0.59) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL20055244 0.88 CYP3A4 (0.59) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL754843 0.87 CYP3A4 (0.54) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL19339631 0.87 CYP3A4 (0.61) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL752995 0.87 PRCP (0.50) CYP3A4CYP2C9KCNH2NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed