SCHEMBL7488563

SCHEMBL7488563

COc1ccc2ccc(Oc3ccnc4cc(OC)c(OC)cc34)cc2c1

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 2/20 0.74
PDGFRB P09619 1/20 0.74
FGFR2 P21802 4/20 0.66
EGFR P00533 1/20 0.62
KDR P35968 3/20 0.60
AURKA O14965 1/20 0.60
ABL1 P00519 1/20 0.60
LCK P06239 1/20 0.60
LYN P07948 1/20 0.60
MET P08581 1/20 0.60
TEK Q02763 1/20 0.60
AURKB Q96GD4 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482292 0.97 PDGFRA (0.78) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL3894972 0.92 PDGFRB (0.74) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL2747893 0.90 PDGFRB (0.67) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL2747234 0.90 PDGFRB (0.67) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL7486400 0.87 FGFR2 (0.84) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL2747998 0.86 PDGFRB (0.71) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL3900264 0.86 EGFR (0.74) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL7481076 0.86 EGFR (0.78) PDGFRAPDGFRBFGFR2EGFR
SCHEMBL925876 0.85 PDGFRB (1.00) PDGFRAPDGFRBFGFR2EGFRKDR
SCHEMBL29573413 0.85 PDGFRB (1.00) PDGFRAPDGFRBFGFR2EGFRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US claimed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP claimed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed