SCHEMBL7494699

SCHEMBL7494699

CC(C)(C)OC(=O)n1c(CN2CCNC(=O)C2)cc2cnccc21

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.36
NAMPT P43490 4/20 0.36
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
GRM5 P41594 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
NR1H2 P55055 2/20 0.34
PRKCH P24723 1/20 0.34
PRKCE Q02156 1/20 0.34
GRM2 Q14416 1/20 0.34
CYP11B2 P19099 1/20 0.34
CDK4 P11802 1/20 0.33
CDK6 Q00534 1/20 0.33
CCNK O75909 1/20 0.33
CDK12 Q9NYV4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4397648 0.86 F10 (0.41) NAMPTCYP2C9NR1H2CCNKCDK12
SCHEMBL1652849 0.82 F10 (0.36) NAMPTCYP2C9NR1H2CDK4CDK6
SCHEMBL4385719 0.81 F10 (0.35) NAMPTNR1H2
SCHEMBL27526708 0.81 F10 (0.36) NAMPTCYP2C9NR1H2CCNKCDK12
SCHEMBL27572872 0.81 SCN9A (0.38) SCN9ANAMPTPDCD1CD274KMT2A
SCHEMBL27572855 0.79 F10 (0.36) NAMPTCYP2C9
SCHEMBL1654543 0.79 F10 (0.39) NAMPTCYP2C9NR1H2
SCHEMBL18848182 0.78 NR1H2 (0.40) NAMPTCYP2C9NR1H2
Tert-Butyl Formate SCHEMBL27572856 0.77 F10 (0.42) NAMPTCYP2C9CCNKCDK12
SCHEMBL27108521 0.77 NR1H2 (0.46) NAMPTCYP2C9NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208097-A2 SUBSTITUTED OXOAZAHETEROCYCLYL COMPOUNDS Aventis Pharmaceuticals Inc. (US) 2002-05-29 EP disclosed
WO-2001007436-A2 SUBSTITUTED OXOAZAHETEROCYCLYL COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2001-02-01 WO disclosed