SCHEMBL7498657

SCHEMBL7498657

COc1ccc(C(CCN2CCC(Nc3nc4ccccc4[nH]3)CC2)CN(C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.54
TACR2 P21452 15/20 0.52
USP2 O75604 1/20 0.44
CXCR6 O00574 1/20 0.40
HRH1 P35367 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7500102 0.95 TACR2 (0.53) KCNH2TACR2USP2CXCR6HRH1
SCHEMBL7493414 0.94 TACR2 (0.51) KCNH2TACR2USP2CXCR6HRH1
SCHEMBL7496523 0.94 TACR2 (0.54) KCNH2TACR2USP2
SCHEMBL8459362 0.92 KCNH2 (0.52) KCNH2TACR2
SCHEMBL7491913 0.92 TACR2 (0.52) KCNH2TACR2USP2
SCHEMBL7496478 0.92 TACR2 (0.59) KCNH2TACR2
SCHEMBL7496327 0.91 TACR2 (0.64) TACR2
SCHEMBL7494874 0.90 TACR2 (0.53) KCNH2TACR2USP2
SCHEMBL7533110 0.87 HRH1 (0.54) TACR2HRH1
SCHEMBL8453525 0.87 TACR2 (0.40) KCNH2TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888336-B1 NOVEL SUBSTITUTED N-METHYL-N-(4-(4-(1H-BENZIMIDAZOL-2-YL-AMINO)P IPERIDIN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES AVENTIS PHARMA INC (US) 2002-08-07 EP disclosed
US-5922737-A Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases HOECHST MARION ROUSSEL, INC. (US) 1999-07-13 US disclosed