SCHEMBL7499279

SCHEMBL7499279

O[C@H](CNCc1ccc(Cl)cc1)COc1ccc(-c2onc3cc(F)ccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
KMT2A Q03164 6/20 0.47
MEN1 O00255 5/20 0.47
PIK3CG P48736 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KCNH2 Q12809 2/20 0.40
CACNA1G O43497 1/20 0.40
ALOX5 P09917 1/20 0.40
ALOX5AP P20292 1/20 0.40
DNM1 Q05193 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1384570 0.94 NPC1 (0.57) NPC1KMT2AMEN1DNM1
SCHEMBL1384566 0.94 NPC1 (0.57) NPC1KMT2AMEN1DNM1
SCHEMBL7493743 0.91 NPC1 (0.48) NPC1KMT2AMEN1KCNH2
SCHEMBL7487764 0.91 MEN1 (0.51) NPC1KMT2AMEN1
SCHEMBL1385112 0.90 NPC1 (0.44) NPC1KMT2AMEN1PIK3CGMAPT
SCHEMBL1385116 0.90 NPC1 (0.44) NPC1KMT2AMEN1PIK3CGMAPT
SCHEMBL7488509 0.86 NPC1 (0.45) NPC1KMT2AMEN1
SCHEMBL1384202 0.86 NPC1 (0.45) NPC1KMT2AMEN1
SCHEMBL7496514 0.86 NPC1 (0.40) NPC1KMT2AMEN1ALOX5ALOX5AP
SCHEMBL1384208 0.86 NPC1 (0.45) NPC1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed