SCHEMBL7500392

SCHEMBL7500392

CCc1cccc(CC)c1CNc1cccn2c(C)c(C)nc12

nearest known ligand 0.88

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 19/20 0.88
CYP2C9 P11712 19/20 0.88
CYP2D6 P10635 10/20 0.88
CYP2C19 P33261 8/20 0.88
CYP1A2 P05177 7/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6062184 0.94 CYP3A4 (1.00) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6352082 0.88 CYP3A4 (0.73) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6351492 0.85 CYP3A4 (0.81) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6350755 0.84 CYP3A4 (0.67) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL7497337 0.84 CYP3A4 (0.66) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6417257 0.83 CYP3A4 (0.66) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6360269 0.83 CYP3A4 (0.80) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
Hydrochloric Acid SCHEMBL6360648 0.82 CYP3A4 (0.79) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6419022 0.81 CYP3A4 (0.77) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2
SCHEMBL6377895 0.80 CYP3A4 (0.72) CYP3A4CYP2C9CYP2D6CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971920-B1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
US-6265415-B1 ANTIULCER AGENT ASTRAZENECA AB (SE) 2001-07-24 US disclosed
EP-0971920-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION Astra Aktiebolag (SE) 2000-01-19 EP disclosed
WO-1998037080-A1 COMPOUNDS FOR INHIBITION OF GASTRIC ACID SECRETION ASTRA AKTIEBOLAG (SE) 1998-08-27 WO disclosed