SCHEMBL7500588

SCHEMBL7500588

COc1ccc(NC(=S)CC(=O)COc2cc(C(=O)Nc3ccc(-c4ncc[nH]4)c(C(F)(F)F)c3)ccc2F)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.45
KDR P35968 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.40
KCNQ3 O43525 3/20 0.39
KCNQ2 O43526 3/20 0.39
KCNE1 P15382 2/20 0.39
KCNQ1 P51787 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
HTR2A P28223 1/20 0.38
POLB P06746 1/20 0.38
ABL1 P00519 3/20 0.38
CXCR1 P25024 1/20 0.38
CXCR2 P25025 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495534 0.83 BRAF (0.42) BRAFKDRSMN1; SMN2MEN1KMT2A
SCHEMBL6846615 0.82 MAPT (0.40) BRAFSMN1; SMN2KCNQ3KCNQ2KCNE1
SCHEMBL7489900 0.80 BRAF (0.44) BRAFKDRKCNQ3KCNQ2KCNE1
SCHEMBL7500274 0.78 BRAF (0.49) BRAFKDRSMN1; SMN2KCNQ3KCNQ2
SCHEMBL7493279 0.75 CYP11B1 (0.51) BRAFKDRABL1
SCHEMBL14083081 0.69 TRPV1 (0.60) SMN1; SMN2MEN1KMT2AMAPTPOLB
SCHEMBL14084122 0.69 TRPV1 (0.59) SMN1; SMN2KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL6846684 0.68 TP53 (0.48) BRAFSMN1; SMN2MAPT
SCHEMBL6841384 0.67 ABL1 (0.41) BRAFSMN1; SMN2MEN1KMT2AMAPT
SCHEMBL14083282 0.65 TRPV1 (0.58) SMN1; SMN2KCNQ3KCNQ2KCNE1KCNQ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252146-A1 AMIDE COMPOUNDS FOR INHIBITING PROTEIN KINASES AGOURON PHARMACEUTICALS, INC. (US) 2002-10-30 EP disclosed
WO-2001053274-A1 AMIDE COMPOUNDS FOR INHIBITING PROTEIN KINASES AGOURON PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed