SCHEMBL7500834

SCHEMBL7500834

Oc1cccc(-c2cc3c(Nc4cccc(Cl)c4)ncnc3[nH]2)c1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.58
ABL1 P00519 4/20 0.58
CDK1 P06493 2/20 0.58
SRC P12931 2/20 0.58
TTBK1 Q5TCY1 3/20 0.55
TTBK2 Q6IQ55 2/20 0.55
PRKCA P17252 1/20 0.54
BRAF P15056 4/20 0.54
TNNI3K Q59H18 3/20 0.54
RAF1 P04049 1/20 0.53
ABL2 P42684 2/20 0.52
FADS1 O60427 1/20 0.51
ERBB2 P04626 1/20 0.51
LCK P06239 1/20 0.50
EIF2AK2 P19525 1/20 0.49
GSK3B P49841 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7502970 0.99 EGFR (0.57) EGFRABL1CDK1SRCTTBK1
SCHEMBL7498606 0.90 BRAF (0.66) EGFRABL1CDK1SRCTTBK1
Bromide SCHEMBL7498610 0.89 BRAF (0.65) EGFRABL1CDK1SRCTTBK1
SCHEMBL4773624 0.88 EGFR (0.59) EGFRABL1CDK1TTBK1TTBK2
SCHEMBL2461054 0.88 BRAF (0.64) EGFRABL1CDK1SRCTTBK1
SCHEMBL8256959 0.86 EIF2AK2 (0.62) EGFRTTBK1TTBK2BRAFTNNI3K
SCHEMBL27442803 0.86 BRAF (0.62) EGFRABL1CDK1SRCTTBK1
SCHEMBL7491484 0.85 TTBK1 (0.54) EGFRABL1TTBK1TTBK2BRAF
SCHEMBL4770048 0.85 EGFR (0.60) EGFRABL1CDK1SRCTTBK1
SCHEMBL7496440 0.84 ABCG2 (0.53) EGFRTTBK1TTBK2BRAFTNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1100778-C Pyrrolopyrimidines and process for their preparation NOVARTIS CO (CH) 2003-02-05 CN claimed
EP-0836605-B1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 2002-02-06 EP claimed
CN-1194647-A Pyrrolopyrimidines and processes for preparation thereof NOVARTIS CO (CH) 1998-09-30 CN claimed
EP-0836605-A1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF Novartis AG (CH) 1998-04-22 EP claimed
WO-1997002266-A1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 1997-01-23 WO claimed