SCHEMBL7500940

SCHEMBL7500940

CC(=O)OCN1C(=O)C(c2cn(C)c3ccccc23)=C(c2cn(C)c3cc([N+](=O)[O-])ccc23)C1=O

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 4/20 0.46
CDK9 P50750 4/20 0.46
CDK2 P24941 3/20 0.42
CCNA2 P20248 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6956384 0.91 CCNT1 (0.46) CCNT1CDK9CDK2CCNA2
SCHEMBL6947835 0.90 CCNT1 (0.44) CCNT1CDK9CDK2CCNA2
SCHEMBL7508601 0.89 CCNT1 (0.47) CCNT1CDK9CDK2CCNA2
SCHEMBL6954175 0.88 CCNT1 (0.43) CCNT1CDK9CDK2CCNA2
SCHEMBL7164524 0.88 CCNT1 (0.47) CCNT1CDK9CDK2CCNA2
Hydrochloric Acid SCHEMBL6954170 0.87 CCNT1 (0.42) CCNT1CDK9CDK2CCNA2
SCHEMBL6950505 0.87 CCNT1 (0.42) CCNT1CDK9CDK2CCNA2MEN1
SCHEMBL7134999 0.87 CDK2 (0.42) CCNT1CDK9CDK2CCNA2
SCHEMBL6948115 0.87 CCNT1 (0.41) CCNT1CDK9CDK2CCNA2MEN1
SCHEMBL6951202 0.87 CCNT1 (0.43) CCNT1CDK9CDK2CCNA2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1155595-C Substituted pyrroles as antiproliferative agents for the treatment of cancer - 2004-06-30 CN disclosed
CN-1378545-A Substituted pyrroles as antiproliferative agents for treatment of cancer HOFFMANN LA ROCHE (CH) 2002-11-06 CN disclosed
EP-1224181-A1 SUBSTITUTED PYRROLES AS ANTIPROLIFERATIVE AGENTS FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001027106-A1 SUBSTITUTED PYRROLES AS ANTIPROLIFERATIVE AGENTS FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2001-04-19 WO disclosed