SCHEMBL750105

SCHEMBL750105

C#Cc1ccc2nc(C3CCCN3C(=O)O)[nH]c2c1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.47
HCRTR2 O43614 19/20 0.47
USP30 Q70CQ3 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2706317 0.86 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL203894 0.86 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL752120 0.85 HCRTR1 (0.45) HCRTR1HCRTR2USP30
SCHEMBL17644204 0.85 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL1293347 0.83 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL19385344 0.81 USP30 (0.66) HCRTR1HCRTR2USP30
SCHEMBL19385343 0.81 USP30 (0.66) HCRTR1HCRTR2USP30
SCHEMBL13494179 0.80 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL2512532 0.80 HTR2B (0.50) HCRTR1HCRTR2
SCHEMBL934057 0.80 CYP3A4 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed