SCHEMBL7501151

SCHEMBL7501151

Cn1cncc1C(=O)Cc1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.46
NPC1 O15118 4/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
PIK3CA P42336 2/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP11B1 P15538 3/20 0.41
CYP11B2 P19099 3/20 0.41
P2RX7 Q99572 1/20 0.40
IDO1 P14902 1/20 0.39
CNR2 P34972 2/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TRPA1 O75762 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501432 0.81 CYP11B1 (0.56) CYP11B1CYP11B2
SCHEMBL10726476 0.79 CTBP2 (0.39) CYP11B1CYP11B2P2RX7IDO1SMN1; SMN2
SCHEMBL10726042 0.79 CTBP2 (0.39) CYP11B1CYP11B2P2RX7IDO1SMN1; SMN2
SCHEMBL10721467 0.77 CYP11B1 (0.38) RAB9AMEN1KMT2ACYP3A4CYP11B1
SCHEMBL10721473 0.77 CYP11B1 (0.38) RAB9AMEN1KMT2ACYP3A4CYP11B1
SCHEMBL3369458 0.76 HTT (0.55) RAB9ANPC1HPGDMAPK1IDO1
SCHEMBL10725110 0.73 CYP11B1 (0.36) RAB9ANPC1L3MBTL1MAPTMEN1
SCHEMBL10725109 0.73 CYP11B1 (0.36) RAB9ANPC1L3MBTL1MAPTMEN1
SCHEMBL20759409 0.73 PREP (0.36) CYP3A4CYP11B1CYP11B2IDO1LMNA
SCHEMBL8916921 0.73 PREP (0.36) MEN1KMT2ACYP3A4MAPK1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020156113-A1 Farnesyl transferase inhibitors; anticancer agents LES LABORATOIRES SERVIER (FR) 2002-10-24 US disclosed
WO-2002057257-A1 CYCLO`C!AZEPANE DERIVATIVES WHICH ARE USED AS FARNESYLTRANSFERASE INHIBITORS AND METHOD FOR THE PREPARATION THEREFOR LES LABORATOIRES SERVIER (FR) 2002-07-25 WO disclosed
WO-2002057258-A1 CYCLO`D!AZEPANE DERIVATIVES WHICH ARE USED AS FARNESYLTRANSFERASE INHIBITORS AND METHOD FOR THE PREPARATION THEREOF LES LABORATOIRES SERVIER (FR) 2002-07-25 WO disclosed
EP-1225170-A2 Cycloheptene compounds, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier S.A. (FR) 2002-07-24 EP disclosed
EP-0216424-A1 Imidazoles, their preparation and their use as fungicides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1987-04-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020156113-A1 Farnesyl transferase inhibitors; anticancer agents COASY, FNTA, FNTB RAB9A 755/4885NPC1 30/4885L3MBTL1 1431/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.