SCHEMBL7505502

SCHEMBL7505502

COC(=O)Oc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5ccccc5)cc4)c3c2)o1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 15/20 0.63
EGFR P00533 12/20 0.63
ERBB4 Q15303 2/20 0.54
CHEK2 O96017 1/20 0.54
ROS1 P08922 1/20 0.54
FLT3 P36888 1/20 0.54
AURKB Q96GD4 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
MKNK2 Q9HBH9 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7506501 0.92 ERBB2 (0.64) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL16575227 0.90 ERBB2 (0.70) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL6768285 0.88 ERBB2 (0.67) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL6763978 0.88 ERBB2 (0.66) ERBB2EGFRERBB4CHEK2ROS1
Hydrochloric Acid SCHEMBL6766485 0.87 ERBB2 (0.65) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL7508142 0.85 EGFR (0.73) ERBB2EGFR
SCHEMBL2999764 0.82 ERBB2 (0.68) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL6767139 0.82 ERBB2 (0.79) ERBB2EGFR
SCHEMBL3320672 0.82 ERBB2 (0.70) ERBB2EGFRERBB4CHEK2ROS1
Hydrochloric Acid SCHEMBL3319025 0.81 ERBB2 (0.67) ERBB2EGFRERBB4CHEK2ROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912559-B1 FUSED HETEROCYCLIC COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LTD (GB) 2002-11-06 EP claimed