SCHEMBL751217

SCHEMBL751217

COC(=O)NCC(C)CC(=O)N1CCCC1c1ncc(-c2ccc(-c3ccc4nc(C5CCCN5C(=O)C(NC(=O)OC)C(C)C)[nH]c4c3)cc2)[nH]1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.68
CYP2C9 P11712 4/20 0.68
NR1I2 O75469 2/20 0.68
KCNH2 Q12809 2/20 0.68
ABCB11 O95342 1/20 0.68
OPRK1 P41145 1/20 0.68
CYP1A2 P05177 2/20 0.64
CYP2D6 P10635 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL751430 1.00 CYP3A4 (0.68) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL13291733 0.92 CYP3A4 (0.71) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL751668 0.91 CYP3A4 (0.72) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL752344 0.91 CYP3A4 (0.55) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL15462358 0.91 CYP3A4 (0.81) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL15462359 0.91 CYP3A4 (0.81) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL2449665 0.91 CYP3A4 (0.81) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL2706507 0.91 CYP3A4 (0.81) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL10177276 0.91 CYP3A4 (0.81) CYP3A4CYP2C9NR1I2KCNH2ABCB11
SCHEMBL14841799 0.91 CYP3A4 (0.81) CYP3A4CYP2C9NR1I2KCNH2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed