SCHEMBL7517017

SCHEMBL7517017

CC1(C)[C@H](C(=O)N[C@@H](Cc2ccc(NC(=O)c3cc(C(F)(F)F)ccc3Cl)cc2)C(=O)O)CC[C@]1(C)C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.59
ITGA4 P13612 11/20 0.59
JAK2 O60674 1/20 0.43
JAK1 P23458 1/20 0.43
TYK2 P29597 1/20 0.43
FPR2 P25090 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PPARG P37231 1/20 0.41
CRHR1 P34998 2/20 0.41
PTGES O14684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098702 1.00 ITGB1 (0.59) ITGB1ITGA4JAK2JAK1TYK2
SCHEMBL7098699 1.00 ITGB1 (0.59) ITGB1ITGA4JAK2JAK1TYK2
SCHEMBL7098046 0.94 ITGB1 (0.51) ITGB1ITGA4JAK2JAK1TYK2
SCHEMBL7098043 0.94 ITGB1 (0.51) ITGB1ITGA4JAK2JAK1TYK2
SCHEMBL7103726 0.91 ITGB1 (0.49) ITGB1ITGA4FPR2MEN1KMT2A
SCHEMBL7103727 0.91 ITGB1 (0.49) ITGB1ITGA4FPR2MEN1KMT2A
SCHEMBL7102565 0.90 ITGB1 (0.48) ITGB1ITGA4MEN1KMT2ANPSR1
SCHEMBL7102563 0.90 ITGB1 (0.48) ITGB1ITGA4MEN1KMT2ANPSR1
SCHEMBL7103673 0.88 ITGB1 (0.59) ITGB1ITGA4
SCHEMBL7104189 0.87 ITGB1 (0.44) ITGB1ITGA4MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991619-A1 INHIBITORS OF $g(a) 4?$g(b) 1?MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 2000-04-12 EP disclosed
WO-1998058902-A1 INHIBITORS OF α4β1MEDIATED CELL ADHESION TANABE SEIYAKU CO., LTD. (JP) 1998-12-30 WO disclosed