SCHEMBL752166

SCHEMBL752166

COC(=O)NCC(C)CC(=O)N1C2CCC(C2)C1c1ncc(-c2ccc3cc(-c4ccc(-c5cnc(C6CC7(CC7)CN6C(=O)C(NC(=O)OC)C(C)C)[nH]5)cc4)ccc3c2)[nH]1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.48
CYP2C9 P11712 6/20 0.48
KCNH2 Q12809 3/20 0.48
NR1I2 O75469 2/20 0.48
ABCB11 O95342 1/20 0.48
OPRK1 P41145 1/20 0.48
CYP1A2 P05177 3/20 0.47
CYP2D6 P10635 2/20 0.45
F2 P00734 1/20 0.30
F11 P03951 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL751153 0.95 CYP3A4 (0.47) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL13465072 0.93 CYP3A4 (0.51) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL20055423 0.93 CYP3A4 (0.51) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL15500334 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL21896824 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL18462755 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL15429815 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL21896686 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL20055161 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11
SCHEMBL2708871 0.91 CYP3A4 (0.55) CYP3A4CYP2C9KCNH2NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed