SCHEMBL7522722

SCHEMBL7522722

COc1cc(C=CC(O)C#N)cc(OC)c1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.51
BCR P11274 1/20 0.51
CYP3A4 P08684 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2B6 P20813 2/20 0.50
CYP2D6 P10635 1/20 0.50
PKM P14618 1/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
TUBB1 Q9H4B7 1/20 0.47
EGFR P00533 4/20 0.46
MAPT P10636 3/20 0.46
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 2/20 0.46
LMNA P02545 2/20 0.46
HPGD P15428 2/20 0.46
BLM P54132 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562829 0.81 ABL1 (0.59) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL9967714 0.79 ABL1 (0.61) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL11301276 0.77 ABL1 (0.54) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL17843663 0.76 ABL1 (0.80) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL16372856 0.76 ABL1 (0.80) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL9123339 0.76 ABL1 (0.58) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL9123345 0.76 ABL1 (0.58) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL5016906 0.75 TUBB1 (0.56) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL5016909 0.75 TUBB1 (0.56) ABL1BCRCYP3A4CYP1A2CYP2C9
SCHEMBL15397238 0.73 ABL1 (0.54) ABL1BCRCYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218370-A2 QUINOLYL PROPYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS Aventis Pharma S.A. (FR) 2002-07-03 EP disclosed
WO-2001025227-A2 QUINOLYL PROPYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS AVENTIS PHARMA S.A. (FR) 2001-04-12 WO disclosed