SCHEMBL7530128

SCHEMBL7530128

COc1ccc(N[C]=O)cc1OC1CCCC1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.62
PDE4A P27815 10/20 0.55
PDE4B Q07343 11/20 0.52
PDE4D Q08499 10/20 0.52
PDE4C Q08493 9/20 0.52
PDE5A O76074 1/20 0.51
PDE1A P54750 1/20 0.51
PDE1B Q01064 1/20 0.51
PDE1C Q14123 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12195758 0.82 POLB (0.64) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL1486262 0.81 SMN1; SMN2 (0.50)
SCHEMBL1157478 0.80 POLB (0.59) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL4193485 0.78 POLB (0.60) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL7358310 0.78 POLB (0.60) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL7338297 0.78 PDE4A (0.55) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL1157367 0.77 PDE4A (0.62) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL1157433 0.77 POLB (0.59) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL1157362 0.77 PDE5A (0.66) POLBPDE4APDE4BPDE4DPDE4C
SCHEMBL1157756 0.77 POLB (0.55) POLBPDE4APDE4BPDE4DPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed