SCHEMBL7538951

SCHEMBL7538951

CN1CCCN(CCN(C)c2ccc(-c3nc4c(OC(N)=O)cccc4[nH]3)cn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.47
DHODH Q02127 4/20 0.45
AURKB Q96GD4 5/20 0.45
AURKA O14965 3/20 0.45
PARP2 Q9UGN5 3/20 0.41
KDR P35968 3/20 0.40
DRD3 P35462 1/20 0.39
PRKD3 O94806 1/20 0.38
PIM1 P11309 1/20 0.38
SRC P12931 1/20 0.38
FLT4 P35916 1/20 0.38
CLK2 P49760 1/20 0.38
GSK3A P49840 1/20 0.38
DYRK1A Q13627 1/20 0.38
PIM3 Q86V86 1/20 0.38
PRKD2 Q9BZL6 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
STK17A Q9UEE5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590927 0.95 AURKB (0.47) PARP1DHODHAURKBAURKAPARP2
SCHEMBL6588412 0.94 AURKB (0.46) PARP1DHODHAURKBAURKAPARP2
SCHEMBL6587813 0.91 AURKB (0.52) PARP1DHODHAURKBAURKAKDR
SCHEMBL6585544 0.90 PARP1 (0.44) PARP1DHODHAURKBAURKAPARP2
SCHEMBL6591730 0.90 AURKB (0.44) PARP1DHODHAURKBAURKAPARP2
SCHEMBL6586442 0.89 AURKB (0.49) PARP1DHODHAURKBAURKAKDR
SCHEMBL6588575 0.88 AURKB (0.54) PARP1DHODHAURKBAURKAKDR
SCHEMBL6800793 0.88 PARP1 (0.63) PARP1DHODHAURKBAURKAPARP2
SCHEMBL6589397 0.87 AURKB (0.51) PARP1DHODHAURKBAURKAKDR
SCHEMBL6588091 0.87 AURKB (0.51) PARP1DHODHAURKBAURKAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed