SCHEMBL7542571

SCHEMBL7542571

CCCN1CCN(c2ccc(C(=O)NCCCCCCCCCCCCCCBr)cn2)CC1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 7/20 0.50
DRD4 P21917 5/20 0.50
DRD2 P14416 5/20 0.50
HTR1A P08908 4/20 0.48
ADRA1D P25100 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
SLC6A4 P31645 1/20 0.48
HTR2A P28223 2/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HDAC6 Q9UBN7 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548525 1.00 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7549534 1.00 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7549515 1.00 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7541225 1.00 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7547128 0.95 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7549536 0.95 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7542767 0.95 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7549212 0.95 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7548225 0.95 DRD3 (0.50) DRD3DRD4DRD2HTR1AADRA1D
SCHEMBL7546434 0.92 HDAC6 (0.52) DRD3DRD4DRD2HTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885886-B1 PYRIDINECARBOXAMIDE DERIVATIVES NISSHIN SEIFUN GROUP INC (JP) 2002-05-29 EP disclosed
US-5972943-A N-(NITRIC ACID,C14-18 ALKYL ESTER)-6-(1-(OPTIONALLY 4-SUBSTITUTED PIPERAZINYL)) PYRIDINE-3-CARBOXAMIDES; METHOD OF SYNTHESIS; ADMINISTERING TO TREAT CEREBRAL EDEMA; NO HYPOTENSIVE SIDE EFFECT NISSHIN FLOUR MILLING CO., LTD. (JP) 1999-10-26 US disclosed
EP-0885886-A1 NOVEL PYRIDINECARBOXAMIDE DERIVATIVES Nisshin Flour Milling Co., Ltd. (JP) 1998-12-23 EP disclosed