SCHEMBL7543878

SCHEMBL7543878

Oc1ccc(N2CCC(O)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.50
TDP1 Q9NUW8 1/20 0.46
CDK1 P06493 1/20 0.45
CDK2 P24941 1/20 0.45
WDR91 A4D1P6 3/20 0.44
ME3 Q16798 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
NOTUM Q6P988 3/20 0.41
ABL1 P00519 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
RORC P51449 3/20 0.40
ESR2 Q92731 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4536703 0.89 TDP1 (0.44) ARTDP1CDK2ME3KDM4E
SCHEMBL2958737 0.88 TDP1 (0.53) TDP1CDK1CDK2ME3KDM4E
SCHEMBL1750887 0.82 AR (0.49) ARCDK1CDK2WDR91ALDH1A1
SCHEMBL1750888 0.82 AR (0.49) ARCDK1CDK2WDR91ALDH1A1
SCHEMBL6365465 0.82 AR (0.49) ARCDK1CDK2WDR91NOTUM
SCHEMBL16695637 0.82 NOTUM (0.60) ARCDK1CDK2WDR91ALDH1A1
SCHEMBL9106437 0.82 NOTUM (0.60) ARCDK1CDK2WDR91ALDH1A1
SCHEMBL15570454 0.82 AR (0.49) ARCDK1CDK2WDR91ALDH1A1
SCHEMBL853367 0.82 AR (0.49) ARTDP1CDK1CDK2WDR91
SCHEMBL33623 0.82 AR (0.49) ARTDP1CDK1CDK2WDR91

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853079-B1 Production of keto acids CIBA SC HOLDING AG (CH) 2002-06-05 EP claimed
US-5925787-A Production of keto acids CIBA SPECIALTY CHEMICALS CORPORATION (US) 1999-07-20 US claimed
EP-0853079-A1 Production of keto acids Ciba SC Holding AG (CH) 1998-07-15 EP claimed
EP-0133578-B1 3-ARYL-3-PYRROLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND MEDICAMENTS CONTAINING THEM FOR THE TREATMENT OF HEART AND VASCULAR DISEASES GÖDECKE AKTIENGESELLSCHAFT (DE) 1990-08-01 EP disclosed
US-4626546-A ANTIISCHEMIC, HYPERTENSIVE AGENTS WARNER-LAMBERT COMPANY (US) 1986-12-02 US disclosed
EP-0133578-A2 3-Aryl-3-pyrroline derivatives, process for their preparation, and medicaments containing them for the treatment of heart and vascular diseases GÖDECKE AKTIENGESELLSCHAFT (DE) 1985-02-27 EP disclosed