SCHEMBL7544381

SCHEMBL7544381

NC1CC(OCc2ccc(-c3nc4ccccc4o3)cc2)CCC1O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
HSD17B10 Q99714 2/20 0.50
TP53 P04637 1/20 0.50
BCHE P06276 1/20 0.45
RAB9A P51151 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
ACSL1 P33121 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7544377 1.00 NPC1 (0.50) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7537523 0.86 NPC1 (0.53) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7537518 0.86 NPC1 (0.53) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7537528 0.86 NPC1 (0.53) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7540462 0.85 NPC1 (0.56) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7540466 0.85 NPC1 (0.56) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7545596 0.83 NPC1 (0.52) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL9158655 0.83 NPC1 (0.51) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7537597 0.83 NPC1 (0.51) NPC1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7543162 0.82 NPC1 (0.51) NPC1KDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676960-B1 CYCLOALKYL AMINE BIS-ARYL SQUALENE SYNTHASE INHIBITORS AVENTIS PHARM PROD INC (US) 2002-05-22 EP disclosed
EP-0676960-A4 1995-11-15 EP disclosed
EP-0676960-A1 CYCLOALKYL AMINE BIS-ARYL SQUALENE SYNTHASE INHIBITORS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1995-10-18 EP disclosed
US-5451596-A Cycloalkyl amine bis-aryl squalene synthase inhibitors RHONE POULENC RORER PHARMACEUTICALS INC. (US) 1995-09-19 US disclosed
WO-1994014435-A1 CYCLOALKYL AMINE BIS-ARYL SQUALENE SYNTHASE INHIBITORS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-07-07 WO disclosed