SCHEMBL7545706

SCHEMBL7545706

CC(C)(C)OC(=O)NC(C)(NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
EPHX2 P34913 1/20 0.46
MDM2 Q00987 1/20 0.45
CASP3 P42574 1/20 0.44
MDM4 O15151 2/20 0.44
TP53 P04637 2/20 0.44
FABP5 Q01469 2/20 0.44
FABP7 O15540 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6673476 0.94 KMT2A (0.54) KMT2AEPHX2CASP3MDM4TP53
SCHEMBL4599855 0.83 KMT2A (0.45) KMT2AEPHX2MDM2CASP3MDM4
SCHEMBL29362505 0.83 KMT2A (0.54) KMT2AEPHX2CASP3MDM4TP53
SCHEMBL29503775 0.83 KMT2A (0.54) KMT2AEPHX2CASP3MDM4TP53
SCHEMBL119779 0.83 KMT2A (0.54) KMT2AEPHX2CASP3MDM4TP53
SCHEMBL20603023 0.83 KMT2A (0.49) KMT2AEPHX2MDM2CASP3MDM4
SCHEMBL18614227 0.82 KMT2A (0.46) KMT2AEPHX2MDM2CASP3MDM4
SCHEMBL31437105 0.82 KMT2A (0.46) KMT2AEPHX2MDM2CASP3MDM4
SCHEMBL18614222 0.82 KMT2A (0.46) KMT2AEPHX2MDM2CASP3MDM4
SCHEMBL6647665 0.82 KMT2A (0.53) KMT2AEPHX2CASP3MDM4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462046-B2 NON-THIAZOLIDINEDIONE PPARGAMMA AGONISTS; USEFUL IN MODULATION OF BLOOD GLUCOSE AND THE INCREASE OF INSULIN SENSITIVITY IN MAMMALS ADVANCED SYNTECH, LLC 2002-10-08 US disclosed
US-20020082263-A1 Heterocycle derivatives as PPAR-gamma agonists ADVANCED SYNTECH LLC 2002-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020082263-A1 Heterocycle derivatives as PPAR-gamma agonists PPARG, PPARD, PPARA KMT2A 2543/4885EPHX2 3662/4885MDM2 2162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.