SCHEMBL7552024

SCHEMBL7552024

O=C1NCCn2c(-c3cccc(F)c3)nc3cccc1c32

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.76
KCNH2 Q12809 1/20 0.53
GRM2 Q14416 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12750589 0.92 PARP1 (0.74) PARP1
SCHEMBL7554564 0.88 PARP1 (0.80) PARP1
SCHEMBL6200038 0.88 PARP1 (0.80) PARP1
SCHEMBL13475803 0.88 PARP1 (0.72) PARP1
SCHEMBL7162599 0.87 PARP1 (0.73) PARP1
SCHEMBL831830 0.87 PARP1 (1.00) PARP1
SCHEMBL7553824 0.86 PARP1 (0.79) PARP1
SCHEMBL12750631 0.86 PARP1 (0.76) PARP1
SCHEMBL7165434 0.85 PARP1 (1.00) PARP1
SCHEMBL7156700 0.84 PARP1 (0.73) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222191-A2 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-07-17 EP disclosed
WO-2001023386-A2 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2001-04-05 WO disclosed