SCHEMBL7559394

SCHEMBL7559394

C=CCc1ccccc1-n1cccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.47
NPC1 O15118 1/20 0.47
MPO P05164 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
G6PD P11413 1/20 0.41
KMT2A Q03164 1/20 0.41
NPBWR1 P48145 1/20 0.39
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
PTPN1 P18031 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRA1A P35348 1/20 0.37
CACNA1G O43497 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12481069 0.79 MAPK1 (0.53) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL9706892 0.79 NOTUM (0.39) ALDH1A1MEN1LMNAKMT2AGABRA1
SCHEMBL110394 0.77 NPC1 (0.51) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL20695961 0.77 MAPK1 (0.51) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL21516008 0.77 MAPK1 (0.51) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL18584960 0.77 NPC1 (0.56) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL4341886 0.75 MAPK1 (0.67) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL20773519 0.75 NPC1 (0.49) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL30288591 0.75 NPC1 (0.49) MAPK1NPC1MPOALDH1A1KDM4E
SCHEMBL30332519 0.75 NPC1 (0.49) MAPK1NPC1MPOALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772598-B1 PREPARATION OF HETEROCYCLIC- AND CARBOCYCLIC-SUBSTITUTED BENZOIC ACIDS MONSANTO TECHNOLOGY LLC (US) 2002-02-06 EP disclosed
EP-0772598-A1 HETEROCYCLIC- AND CARBOCYCLIC-SUBSTITUTED BENZOIC ACIDS AND SYNTHESIS THEREOF MONSANTO COMPANY (US) 1997-05-14 EP disclosed
US-5587485-A CATALYTIC OXIDATION OF THE CORRESPONDING ALKYL SUBSTITUTED BENZENE COMPOUND MONSANTO COMPANY (US) 1996-12-24 US disclosed
WO-1996002515-A1 HETEROCYCLIC- AND CARBOCYCLIC-SUBSTITUTED BENZOIC ACIDS AND SYNTHESIS THEREOF MONSANTO COMPANY (US) 1996-02-01 WO disclosed