SCHEMBL7560175

SCHEMBL7560175

COc1ccc2nccc(CCCC3CCN(CCCc4ccccc4)CC3CO)c2c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 2/20 0.53
KCNH2 Q12809 7/20 0.48
GRIN1 Q05586 2/20 0.45
GRIN2B Q13224 2/20 0.45
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7466144 1.00 CCR8 (0.53) CCR8KCNH2GRIN1GRIN2BGAA
Oxalic Acid SCHEMBL7728019 0.97 CCR8 (0.52) CCR8KCNH2GRIN1GRIN2B
SCHEMBL7455480 0.92 CCR8 (0.53) CCR8KCNH2KDM4EALDH1A1MAPT
SCHEMBL7725846 0.91 CCR8 (0.53) CCR8KCNH2
SCHEMBL7724893 0.91 CCR8 (0.52) CCR8KCNH2
SCHEMBL7724897 0.91 CCR8 (0.52) CCR8KCNH2
SCHEMBL7728026 0.90 CCR8 (0.52) CCR8KCNH2
SCHEMBL7731901 0.90 CCR8 (0.51) CCR8KCNH2KDM4EALDH1A1MAPT
SCHEMBL7462927 0.89 CCR8 (0.54) CCR8KCNH2
SCHEMBL7724509 0.89 CCR8 (0.51) CCR8KCNH2GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218370-A2 QUINOLYL PROPYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS Aventis Pharma S.A. (FR) 2002-07-03 EP disclosed
US-6403610-B1 ANTIMICROBIAL AGENTS AVENTIS PHARMA S.A. (FR) 2002-06-11 US disclosed
WO-2001025227-A2 QUINOLYL PROPYL PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS AVENTIS PHARMA S.A. (FR) 2001-04-12 WO disclosed