SCHEMBL756283

SCHEMBL756283

[CH2]c1cc(N2C(=O)C(C)(C)Oc3cc(NS(C)(=O)=O)cc(F)c32)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 6/20 0.53
AR P10275 1/20 0.35
BRD4 O60885 4/20 0.34
PGR P06401 1/20 0.32
HAVCR2 Q8TDQ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL755980 0.89 NR3C2 (0.56) NR3C2ARBRD4PGR
SCHEMBL754215 0.87 NR3C2 (0.61) NR3C2ARBRD4PGR
SCHEMBL756053 0.86 NR3C2 (0.51) NR3C2ARBRD4
SCHEMBL754664 0.86 NR3C2 (0.59) NR3C2ARBRD4PGR
SCHEMBL754681 0.85 NR3C2 (0.53) NR3C2ARPGR
SCHEMBL755391 0.85 NR3C2 (0.72) NR3C2ARBRD4PGR
SCHEMBL758564 0.84 NR3C2 (0.69) NR3C2BRD4PGR
SCHEMBL756893 0.82 NR3C2 (0.55) NR3C2ARBRD4
SCHEMBL755896 0.82 AR (0.58) NR3C2AR
SCHEMBL755535 0.82 NR3C2 (0.54) NR3C2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984345-B9 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORP (JP) 2012-03-21 EP claimed
EP-1984345-B1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORP (JP) 2011-08-31 EP claimed