SCHEMBL7563757

SCHEMBL7563757

N#Cc1cnc2cnc(Nc3ccccc3)cc2c1Nc1cccc(Br)c1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.71
ERBB2 P04626 15/20 0.71
GAK O14976 1/20 0.64
MAP2K1 Q02750 1/20 0.53
MAP3K8 P41279 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6644272 0.90 EGFR (0.69) EGFRERBB2GAK
SCHEMBL6642786 0.86 EGFR (0.70) EGFRERBB2GAK
SCHEMBL6646331 0.84 EGFR (0.70) EGFRERBB2GAK
SCHEMBL6643911 0.84 EGFR (0.70) EGFRERBB2GAK
SCHEMBL27459387 0.83 EGFR (0.72) EGFRERBB2GAKMAP2K1
SCHEMBL6644226 0.83 EGFR (0.69) EGFRERBB2GAK
SCHEMBL6381329 0.83 EGFR (1.00) EGFRERBB2GAK
SCHEMBL1893339 0.80 EGFR (0.70) EGFRERBB2GAK
SCHEMBL4769778 0.79 EGFR (0.68) EGFRERBB2GAKMAP2K1MAP3K8
SCHEMBL6647860 0.79 EGFR (0.62) EGFRERBB2GAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020165229-A1 Substituted 3-cyano-[1.7], [1.5], and [1.8] naphthyridine inhibitors of tyrosine kinases AMERICAN CYANAMID COMPANY 2002-11-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020165229-A1 Substituted 3-cyano-[1.7], [1.5], and [1.8] naphthyridine inhibitors of tyrosine kinases ABL1, ROS1, ALK EGFR 14/4885ERBB2 4/4885GAK 354/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.