SCHEMBL7567907

SCHEMBL7567907

CCOC(=O)ON1CCNCC1C(=O)c1cc(NS(=O)(=O)c2ccc3c(c2)OCO3)c(Oc2ccccc2OC)c(OCCO)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 8/20 0.42
EDNRB P24530 4/20 0.37
GLRA3 O75311 2/20 0.35
GLRB P48167 2/20 0.35
POLB P06746 1/20 0.34
ALDH1A1 P00352 3/20 0.34
USP2 O75604 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
MAPT P10636 1/20 0.34
ABCC3 O15438 1/20 0.34
ABCC4 O15439 1/20 0.34
NR1I2 O75469 1/20 0.34
ABCB11 O95342 1/20 0.34
DHPS P49366 1/20 0.34
NR1H3 Q13133 1/20 0.34
NR1I3 Q14994 1/20 0.34
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570858 0.81 EDNRA (0.48) EDNRAEDNRBPOLBALDH1A1
SCHEMBL7567975 0.80 EDNRA (0.55) EDNRAEDNRBGLRA3GLRBALDH1A1
SCHEMBL7567961 0.80 EDNRA (0.55) EDNRAEDNRBGLRA3GLRBPOLB
SCHEMBL7570509 0.78 EDNRA (0.49) EDNRAEDNRBPOLBALDH1A1SMN1; SMN2
SCHEMBL7569569 0.78 EDNRA (0.52) EDNRAEDNRBALDH1A1USP2HSP90AA1
SCHEMBL7567923 0.78 EDNRA (0.52) EDNRAEDNRBGLRA3GLRBALDH1A1
SCHEMBL7567596 0.76 EDNRA (0.50) EDNRAEDNRBGLRA3GLRBALDH1A1
SCHEMBL7567694 0.73 EDNRA (0.60) EDNRAEDNRB
SCHEMBL7568711 0.71 EDNRA (0.62) EDNRAEDNRB
SCHEMBL7569450 0.71 EDNRB (0.53) EDNRAEDNRBALDH1A1MAPTABCC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799206-B1 ARYL- AND HETARYL-SULFONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ENDOTHELIN ANTAGONISTS HOFFMANN LA ROCHE (CH) 2002-09-11 EP claimed