SCHEMBL7577005

SCHEMBL7577005

Cc1cc(C2C(=O)N(C)C(=N)N[C@]2(C)c2cccc(C#N)c2)ccc1C#N

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.36
BACE2 Q9Y5Z0 2/20 0.32
PGR P06401 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GSK3A P49840 2/20 0.31
NSD2 O96028 1/20 0.31
PAX8 Q06710 1/20 0.31
CTSD P07339 1/20 0.31
HSD11B1 P28845 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202597 1.00 BACE1 (0.36) BACE1BACE2PGRALDH1A1GSK3A
SCHEMBL13055205 1.00 BACE1 (0.36) BACE1BACE2PGRALDH1A1GSK3A
SCHEMBL7558336 0.90 BACE1 (0.35) BACE1BACE2PGRALDH1A1NSD2
SCHEMBL13054464 0.90 BACE1 (0.35) BACE1BACE2PGRALDH1A1NSD2
SCHEMBL7557016 0.90 BACE1 (0.39) BACE1BACE2PGRALDH1A1NSD2
SCHEMBL13054247 0.90 BACE1 (0.39) BACE1BACE2PGRALDH1A1NSD2
SCHEMBL14105172 0.89 AR (0.31)
SCHEMBL7574530 0.89 BACE1 (0.39) BACE1BACE2PGRALDH1A1NSD2
SCHEMBL13054721 0.89 BACE1 (0.39) BACE1BACE2PGRALDH1A1NSD2
SCHEMBL7582473 0.88 BACE1 (0.32) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed