SCHEMBL7584511

SCHEMBL7584511

Cc1ccccc1Nc1ccc(C(=NO)c2c(C)noc2C)c(Cl)c1.Cn1ccnc1C(=NO)c1ccc(Nc2ccccc2N)cc1Cl.Cn1ccnc1C(=NO)c1ccc(Nc2ccccc2[N+](=O)[O-])cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.45
MAPK13 O15264 8/20 0.45
MAPK12 P53778 8/20 0.45
MAPK11 Q15759 8/20 0.45
ALDH1A1 P00352 5/20 0.33
MAPT P10636 5/20 0.33
LMNA P02545 3/20 0.33
GAA P10253 3/20 0.33
KMT2A Q03164 3/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GRM4 Q14833 1/20 0.32
TDP1 Q9NUW8 2/20 0.31
AGTR1 P30556 1/20 0.31
ALKBH5 Q6P6C2 1/20 0.30
FTO Q9C0B1 1/20 0.30
MEN1 O00255 2/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7585243 0.89 MAPK14 (0.37) MAPK14MAPK13MAPK12MAPK11
SCHEMBL7082270 0.85 MAPK13 (0.53) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL7082272 0.85 MAPK13 (0.53) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL7079620 0.81 MAPK14 (0.48) MAPK14MAPK13MAPK12MAPK11MAPT
SCHEMBL7079618 0.81 MAPK14 (0.48) MAPK14MAPK13MAPK12MAPK11MAPT
SCHEMBL7083146 0.79 MAPK14 (0.51) MAPK14MAPK13MAPK12MAPK11GRM4
SCHEMBL7083149 0.79 MAPK14 (0.51) MAPK14MAPK13MAPK12MAPK11GRM4
SCHEMBL7080598 0.78 MAPK14 (0.52) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL7080621 0.78 MAPK14 (0.52) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL7076539 0.74 MAPK13 (0.64) MAPK14MAPK13MAPK12MAPK11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002083622-A2 NOVEL AMINOPHENYL KETONE DERIVATIVES LEO PHARMA A/S (DK) 2002-10-24 WO disclosed