SCHEMBL7585628

SCHEMBL7585628

Nc1cc(Br)c(Cl)c(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.58
MAPT P10636 1/20 0.58
CYP3A4 P08684 3/20 0.45
TP53 P04637 1/20 0.45
ALDH1A1 P00352 4/20 0.43
THRB P10828 1/20 0.39
TSHR P16473 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 1/20 0.33
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
CA4 P22748 1/20 0.31
AHR P35869 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29675989 0.86 CYP3A4 (0.50) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL21050901 0.86 CYP3A4 (0.50) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL26694609 0.82 GAA (0.46) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL21050751 0.82 GAA (0.46) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL12397904 0.77 GAA (0.42) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL5660899 0.77 POLB (0.47) GAAMAPTALDH1A1TSHRMAPK1
SCHEMBL525650 0.75 CYP3A4 (0.65) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL25259748 0.73 TDP1 (0.47) CYP3A4ALDH1A1TSHRCA1CA2
SCHEMBL9323230 0.73 MAPT (0.65) GAAMAPTCYP3A4TP53ALDH1A1
SCHEMBL5076239 0.73 MAPT (1.00) GAAMAPTCYP3A4TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP disclosed
US-6281214-B1 USEFUL FOR TREATING AND AMELIORATING MENTAL DISORDERS EISAI CO., LTD (JP) 2001-08-28 US disclosed
US-5849912-A Biphenyl derivatives EISAI CO., LTD. (JP) 1998-12-15 US disclosed
CN-1117966-A Biphenyl derivatives EISAI CO LTD (JP) 1996-03-06 CN disclosed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP disclosed