SCHEMBL7586563

SCHEMBL7586563

CC1(c2ccc(O)cc2)COc2cc(O)ccc2C1c1cccc(OCCCCCS(=O)(=O)CCCC(F)(F)C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.49
KCNE1 P15382 3/20 0.31
KCNQ1 P51787 3/20 0.31
KCNH2 Q12809 1/20 0.31
ESR2 Q92731 5/20 0.31
CYP3A4 P08684 2/20 0.30
ALOX15 P16050 2/20 0.30
NR1I2 O75469 1/20 0.30
NR3C1 P04150 1/20 0.30
PGR P06401 1/20 0.30
ESRRA P11474 1/20 0.30
EPHX2 P34913 1/20 0.30
PPARG P37231 1/20 0.30
NR1H4 Q96RI1 1/20 0.30
SIRT5 Q9NXA8 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7587903 0.99 ESR1 (0.48) ESR1KCNE1KCNQ1KCNH2ESR2
SCHEMBL7587953 0.88 ESR1 (0.37) ESR1ESR2CYP3A4ALOX15KDM4E
SCHEMBL7589642 0.87 ESR1 (0.36) ESR1ESR2CYP3A4ALOX15KDM4E
SCHEMBL7589074 0.87 ESR1 (0.36) ESR1ESR2CYP3A4ALOX15KDM4E
SCHEMBL7585601 0.86 ESR1 (0.35) ESR1ESR2CYP3A4ALOX15KDM4E
SCHEMBL7585376 0.82 ESR1 (0.43) ESR1ESR2CYP3A4ALOX15NR1I2
SCHEMBL7592604 0.81 ESR1 (0.51) ESR1ESR2PPARG
SCHEMBL5856046 0.81 ESR1 (0.40) ESR1ESR2HDAC6
SCHEMBL5855904 0.81 ESR1 (0.40) ESR1ESR2HDAC6
SCHEMBL5854563 0.81 ESR1 (0.40) ESR1ESR2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944613-B1 BENZOPYRAN DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2002-10-09 EP claimed
EP-0944613-A1 NOVEL BENZOPYRAN DERIVATIVES C & C Research Laboratories (KR) 1999-09-29 EP claimed
WO-1998025916-A1 NOVEL BENZOPYRAN DERIVATIVES C & C RESEARCH LABORATORIES (KR) 1998-06-18 WO claimed
EP-0944613-B1 BENZOPYRAN DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2002-10-09 EP disclosed
US-6153768-A RECEPTOR BLOCKING ANTIESTROGENS HAVING REDUCED SIDE EFFECTS C & C RESEARCH LABORATORIES (KR) 2000-11-28 US disclosed
EP-0944613-A1 NOVEL BENZOPYRAN DERIVATIVES C & C Research Laboratories (KR) 1999-09-29 EP disclosed
WO-1998025916-A1 NOVEL BENZOPYRAN DERIVATIVES C & C RESEARCH LABORATORIES (KR) 1998-06-18 WO disclosed