SCHEMBL7596469

SCHEMBL7596469

COc1cccc(C(=O)NCCN2CCN(C(=O)c3ccc(Cl)c(Cl)c3)CC2)c1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 15/20 0.68
CCR3 P51677 2/20 0.68
DRD2 P14416 5/20 0.66
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
MAPT P10636 1/20 0.65
PMP22 Q01453 1/20 0.65
CYP2C9 P11712 1/20 0.63
CYP2C19 P33261 1/20 0.63
KMT2A Q03164 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6396151 0.99 DRD4 (0.67) DRD4CCR3DRD2CYP1A2CYP3A4
Isobutyramide SCHEMBL27550765 0.93 CCR3 (0.60) DRD4CCR3DRD2CYP1A2CYP3A4
SCHEMBL6396896 0.87 KMT2A (0.65) CCR3MAPTKMT2A
Hydrochloric Acid SCHEMBL27570386 0.85 CCR3 (0.74) DRD4CCR3DRD2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL27570348 0.81 CCR3 (0.71) DRD4CCR3DRD2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL6402140 0.81 CCR3 (0.71) DRD4CCR3DRD2CYP1A2CYP3A4
SCHEMBL5658825 0.81 CCR3 (1.00) DRD4CCR3DRD2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL6399917 0.80 CCR3 (0.98) DRD4CCR3DRD2CYP1A2CYP3A4
SCHEMBL1322020 0.79 DRD4 (1.00) DRD4DRD2CYP1A2CYP3A4CYP2D6
SCHEMBL6399874 0.79 HPGD (0.57) CCR3MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165545-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2002-01-02 EP disclosed
WO-2000058305-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2000-10-05 WO disclosed