SCHEMBL7599776

SCHEMBL7599776

Cc1[nH]cc2c(=O)n(-c3ccc(Cl)cc3)nc-2c1-c1ccc(NCC(C)(C)N)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.34
GAA P10253 7/20 0.34
NPSR1 Q6W5P4 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
AURKA O14965 1/20 0.32
SYK P43405 1/20 0.32
LMNA P02545 2/20 0.32
PSD A5PKW4 1/20 0.32
CNR1 P21554 1/20 0.32
SRC P12931 1/20 0.31
BRAF P15056 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2648050 0.85 CNR1 (0.39) GAAMAPTPOLBTDP1L3MBTL1
SCHEMBL2649657 0.85 GAA (0.44) PTGS2GAANPSR1SMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL2662079 0.84 GAA (0.43) PTGS2GAANPSR1SMN1; SMN2MAPT
SCHEMBL7441207 0.83 JAK1 (0.38) PTGS2GAANPSR1SMN1; SMN2POLB
SCHEMBL2649011 0.82 GAA (0.40) PTGS2GAANPSR1SMN1; SMN2MAPT
SCHEMBL7434904 0.82 GAA (0.38) PTGS2GAANPSR1SMN1; SMN2MAPT
SCHEMBL2650198 0.81 PSD (0.42) PTGS2SMN1; SMN2MAPTPOLBMEN1
SCHEMBL2649301 0.80 MAPT (0.43) GAANPSR1SMN1; SMN2MAPTTDP1
SCHEMBL2650368 0.80 GAA (0.40) PTGS2GAANPSR1SMN1; SMN2MAPT
SCHEMBL2649535 0.80 GAA (0.43) PTGS2GAANPSR1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333336-B1 GAMMA-AMINOBUTYRIC ACID RECEPTORS AS ANTICONVULSANTS FORMING THE COMPOUND BY AMIDATION MERCK SHARP & DOHME LTD. (GB) 2001-12-25 US disclosed