SCHEMBL760030

SCHEMBL760030

C[C@H]1CC2(CCN1CC1CCC1)C(N[C@@H]1CCCC[C@H]1F)=NC(=O)N2c1cccc(F)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.34
BACE2 Q9Y5Z0 1/20 0.33
ADORA3 P0DMS8 2/20 0.32
ADORA1 P30542 2/20 0.32
ADORA2A P29274 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10293318 1.00 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
SCHEMBL755429 1.00 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
SCHEMBL755862 1.00 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
Hydrochloric Acid SCHEMBL757214 0.99 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
Hydrochloric Acid SCHEMBL757169 0.99 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
SCHEMBL754725 0.99 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
SCHEMBL755943 0.99 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
SCHEMBL758021 0.99 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
Hydrochloric Acid SCHEMBL756099 0.98 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A
Hydrochloric Acid SCHEMBL755842 0.98 BACE1 (0.34) BACE1BACE2ADORA3ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910364-B1 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME (US) 2012-03-21 EP disclosed