SCHEMBL7605348

SCHEMBL7605348

CC[Si](CC)(CC)OC(CBr)c1ccc(OCc2ccccc2)c(NS(C)(=O)=O)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.44
TRPV1 Q8NER1 3/20 0.42
ADRB3 P13945 6/20 0.41
NPC1 O15118 1/20 0.40
AR P10275 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
ESRRA P11474 1/20 0.39
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
PRSS1 P07477 1/20 0.38
F7 P08709 1/20 0.38
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7605339 1.00 CYP19A1 (0.44) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL6479480 0.90 CYP19A1 (0.44) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL5483348 0.90 CYP19A1 (0.44) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL4817546 0.90 CYP19A1 (0.44) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL6986483 0.87 ADRB3 (0.48) CYP19A1TRPV1ADRB3PDE4APDE4B
SCHEMBL2454673 0.86 CYP19A1 (0.43) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL14090675 0.86 CYP19A1 (0.43) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL2452164 0.86 CYP19A1 (0.43) CYP19A1TRPV1ADRB3NPC1AR
SCHEMBL7113237 0.82 ADRB3 (0.45) CYP19A1TRPV1ADRB3SMN1; SMN2
SCHEMBL7040215 0.82 ADRB3 (0.61) ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed