SCHEMBL7606040

SCHEMBL7606040

CCOC(=O)CCc1ccc(C#N)c(OCC(O)CNC(C)(C)Cc2ccc3ccccc3c2)c1

nearest known ligand 0.91

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASR P41180 18/20 0.91
CYP2D6 P10635 10/20 0.91
SLC6A2 P23975 8/20 0.91
SLC6A4 P31645 8/20 0.91
SLC6A3 Q01959 8/20 0.91
KCNH2 Q12809 8/20 0.91
ADRB2 P07550 5/20 0.91
ADRB3 P13945 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606034 1.00 CASR (0.91) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7608757 0.99 CASR (0.91) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7608764 0.99 CASR (0.91) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL3355497 0.95 CASR (0.83) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL3355486 0.95 CASR (0.83) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL3355494 0.95 CASR (0.83) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6375455 0.95 CASR (1.00) CASRCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6375430 0.95 CASR (1.00) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7603298 0.95 CASR (0.83) CASRCYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7603308 0.95 CASR (0.83) CASRCYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US claimed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP claimed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP claimed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO claimed
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US disclosed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP disclosed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed