SCHEMBL7608258

SCHEMBL7608258

COc1ccc(CC(C)(C)NC[C@@H](O)COc2ccc(CCCO)cc2)cc1

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASR P41180 18/20 0.75
ADRB2 P07550 6/20 0.60
ADRB3 P13945 5/20 0.60
CYP2D6 P10635 3/20 0.59
SLC6A2 P23975 3/20 0.59
SLC6A4 P31645 3/20 0.59
SLC6A3 Q01959 3/20 0.59
KCNH2 Q12809 3/20 0.59
ADRB1 P08588 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7608752 0.99 CASR (0.73) CASRADRB2ADRB3CYP2D6SLC6A2
SCHEMBL7606721 0.93 CASR (0.78) CASRADRB2ADRB3CYP2D6SLC6A2
SCHEMBL14382960 0.91 CASR (0.90) CASRADRB2ADRB3CYP2D6SLC6A2
Hydrochloric Acid SCHEMBL5509997 0.89 CASR (0.88) CASRADRB2ADRB3CYP2D6SLC6A2
Hydrochloric Acid SCHEMBL5508953 0.87 CASR (0.77) CASRADRB2ADRB3CYP2D6SLC6A2
SCHEMBL14382945 0.86 CASR (1.00) CASRADRB2ADRB3CYP2D6SLC6A2
SCHEMBL14382943 0.86 CASR (1.00) CASRADRB2ADRB3CYP2D6SLC6A2
SCHEMBL14382947 0.86 CASR (1.00) CASRADRB2ADRB3CYP2D6SLC6A2
SCHEMBL14383005 0.85 CASR (0.80) CASRADRB2ADRB3CYP2D6SLC6A2
Hydrochloric Acid SCHEMBL5510007 0.85 CASR (0.80) CASRADRB2ADRB3CYP2D6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US claimed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP claimed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP claimed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO claimed
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US disclosed