SCHEMBL7609129

SCHEMBL7609129

C=CC[C@H]1C[C@H]2[C@@H]3CC=C4N(C)C(=O)CC[C@]4(C)[C@H]3CC[C@]2(C)C1=O

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 2/20 0.54
CYP2C19 P33261 1/20 0.44
CYP19A1 P11511 6/20 0.44
SRD5A2 P31213 2/20 0.41
CYP1B1 Q16678 1/20 0.40
G6PD P11413 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7609134 1.00 SRD5A1 (0.54) SRD5A1CYP2C19CYP19A1SRD5A2CYP1B1
SCHEMBL7711721 0.79 SRD5A1 (0.49) SRD5A1CYP19A1SRD5A2CYP1B1G6PD
SCHEMBL7711725 0.79 SRD5A1 (0.49) SRD5A1CYP19A1SRD5A2CYP1B1G6PD
SCHEMBL7616969 0.78 SRD5A1 (0.51) SRD5A1CYP2C19CYP19A1SRD5A2
SCHEMBL7616961 0.78 SRD5A1 (0.51) SRD5A1CYP2C19CYP19A1SRD5A2
SCHEMBL7609770 0.78 SRD5A1 (0.51) SRD5A1CYP2C19CYP19A1SRD5A2
SCHEMBL7609766 0.78 SRD5A1 (0.51) SRD5A1CYP2C19CYP19A1SRD5A2
SCHEMBL3795654 0.77 SRD5A1 (0.61) SRD5A1CYP19A1G6PD
SCHEMBL7617616 0.77 SRD5A1 (0.61) SRD5A1CYP19A1G6PD
SCHEMBL8065395 0.76 SRD5A1 (0.60) SRD5A1CYP2C19CYP19A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880540-B1 17-BETA-CYCLOPROPYL(AMINO/OXY) 4-AZA STEROIDS AS ACTIVE INHIBITORS OF TESTOSTERONE 5-ALPHA-REDUCTASE AND C17-20-LYASE AVENTIS PHARMA INC (US) 2002-06-12 EP disclosed
US-6365597-B1 FOR THERAPY OF ANDROGEN AND ESTROGEN MEDIATED DISORDERS, INCLUDING BENIGN PROSTATIC HYPERPLASIA, ANDROGEN MEDIATED PROSTATE CANCER, ESTROGEN MEDIATED BREAST CANCER AND ACNE AVENTIS PHARMACEUTICALS INC. 2002-04-02 US disclosed