SCHEMBL7618445

SCHEMBL7618445

CCCN(CCC)CCCOc1cc(NC(=O)C=Cc2ccc(C(C)C)cc2)ccc1OC

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 14/20 0.57
ACHE P22303 13/20 0.57
SLC2A1 P11166 1/20 0.55
TP53 P04637 1/20 0.51
MAPT P10636 1/20 0.51
TRPV1 Q8NER1 1/20 0.51
GCGR P47871 1/20 0.51
HDAC1 Q13547 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651296 0.95 SLC2A1 (0.58) BCHEACHESLC2A1TP53MAPT
SCHEMBL7620255 0.91 BCHE (0.58) BCHEACHESLC2A1TP53MAPT
SCHEMBL7612941 0.89 SLC2A1 (0.66) BCHEACHESLC2A1TP53MAPT
SCHEMBL7612936 0.89 SLC2A1 (0.66) BCHEACHESLC2A1TP53MAPT
SCHEMBL7612949 0.88 BCHE (0.58) BCHEACHESLC2A1TP53MAPT
SCHEMBL7614846 0.87 BCHE (0.56) BCHEACHESLC2A1TP53MAPT
SCHEMBL7612442 0.86 BCHE (0.63) BCHEACHESLC2A1TP53MAPT
SCHEMBL7613897 0.86 BCHE (0.60) BCHEACHESLC2A1TP53MAPT
SCHEMBL7618033 0.86 SLC2A1 (0.73) BCHEACHESLC2A1TP53MAPT
SCHEMBL7651286 0.86 SLC2A1 (0.73) BCHEACHESLC2A1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100495-A4 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORP (US) 2002-09-25 EP disclosed
EP-1100495-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP disclosed
WO-2000006153-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed