SCHEMBL7620529

SCHEMBL7620529

Cc1cc(C(=O)CBr)ccc1Cl.Cc1cc(C(=O)CBr)ccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.55
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
PTPN1 P18031 6/20 0.49
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
TAS1R2 Q8TE23 1/20 0.46
MCL1 Q07820 1/20 0.44
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
GNG2 P59768 1/20 0.41
GNB1 P62873 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL243504 1.00 GSK3B (0.55) GSK3BCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23112482 0.85 GSK3B (0.55) GSK3BCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2278168 0.83 CYP3A4 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19TAS1R3
SCHEMBL2097486 0.83 GSK3B (0.53) GSK3BCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL27778655 0.83 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C9CYP2C19TAS1R3
SCHEMBL1726590 0.82 GSK3B (0.61) GSK3BPTPN1
SCHEMBL30187429 0.82 GSK3B (0.61) GSK3BPTPN1
SCHEMBL29514695 0.82 GSK3B (0.61) GSK3BPTPN1
SCHEMBL747174 0.82 GSK3B (0.61) GSK3BPTPN1
SCHEMBL2075296 0.81 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US disclosed