SCHEMBL7620979

SCHEMBL7620979

Cc1cc(F)cc(C)c1CC(Br)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
SLC6A4 P31645 7/20 0.33
GBA1 P04062 3/20 0.33
SLC6A2 P23975 3/20 0.33
SLC6A3 Q01959 2/20 0.33
TAAR1 Q96RJ0 1/20 0.32
OPRK1 P41145 1/20 0.31
HKDC1 Q2TB90 1/20 0.31
CCR5 P51681 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12466368 0.77 IDO1 (0.41) IDO1TDO2GBA1OPRK1
SCHEMBL5973963 0.74 TDP1 (0.42) IDO1TDO2SLC6A4SLC6A2SLC6A3
SCHEMBL10778612 0.74 SLC6A2 (0.47) SLC6A4SLC6A2SLC6A3TAAR1
SCHEMBL7620984 0.72 TAAR1 (0.37) SLC6A4SLC6A2SLC6A3TAAR1
SCHEMBL28496558 0.67 CNR2 (0.48) IDO1TDO2SLC6A4SLC6A2TAAR1
SCHEMBL27666865 0.67 TAAR1 (0.46) IDO1SLC6A4SLC6A2SLC6A3TAAR1
SCHEMBL1641620 0.66 SLC6A2 (0.48) SLC6A4SLC6A2SLC6A3TAAR1TSHR
SCHEMBL19143212 0.66 CYP19A1 (0.39) SLC6A4SLC6A3
SCHEMBL19317398 0.66 CYP19A1 (0.39) SLC6A4SLC6A3
SCHEMBL25097170 0.64 HRH1 (0.40) IDO1TDO2SLC6A4GBA1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906288-B1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2002-11-06 EP disclosed
US-6465505-B1 SUCH AS 4-(2,6-DIMETHYLBENZYLAMINO OR BENZYLOXY)-2-METHYL BENZIMIDAZOLE; INHIBITING EXOGENOUS OR ENDOGENOUS STIMULATED GASTRIC ACID SECRETION; PREVENTION AND TREATMENT OF GASTRO-INTESTINAL INFLAMMATORY DISEASES ASTRAZENECA AB (SE) 2002-10-15 US disclosed
EP-0906288-A1 NEW COMPOUNDS Astra Aktiebolag (SE) 1999-04-07 EP disclosed
WO-1997047603-A1 NEW COMPOUNDS ASTRA AKTIEBOLAG (SE) 1997-12-18 WO disclosed