SCHEMBL762863

SCHEMBL762863

C=CCN1CC(=O)N2[C@@H](Cc3ccc(NC=O)cc3)C(=O)N(Cc3cccc(C(N)=O)c3)C[C@@H]2N1C(=O)NCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 19/20 0.61
TCF4 P15884 1/20 0.53
CTNNB1 P35222 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2899926 0.92 CYP3A4 (0.68) CYP3A4
SCHEMBL10292458 0.92 CYP3A4 (0.68) CYP3A4
SCHEMBL13028883 0.89 CYP3A4 (0.67) CYP3A4
SCHEMBL10291369 0.88 CYP3A4 (0.58) CYP3A4TCF4CTNNB1
SCHEMBL13028822 0.88 CYP3A4 (0.60) CYP3A4TCF4CTNNB1
SCHEMBL2894885 0.88 CYP3A4 (0.67) CYP3A4
SCHEMBL750416 0.88 CYP3A4 (0.67) CYP3A4
SCHEMBL2894978 0.86 CYP3A4 (0.66) CYP3A4
SCHEMBL13354127 0.86 CYP3A4 (0.61) CYP3A4TCF4CTNNB1
SCHEMBL762363 0.86 CYP3A4 (0.66) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138337-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-03-20 US disclosed
US-8049008-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2011-11-01 US disclosed
US-7671054-B1 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2010-03-02 US disclosed
US-7671054-B1 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2010-03-02 US disclosed