SCHEMBL762894

SCHEMBL762894

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)Cc3ccc(-c4cccnc4OC)cc3)C2)nc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 11/20 0.42
HRH1 P35367 11/20 0.42
CYP2D6 P10635 8/20 0.42
CHRM1 P11229 3/20 0.41
CYP3A4 P08684 1/20 0.39
PROKR1 Q8TCW9 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740659 0.93 HRH1 (0.41) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL740660 0.93 HRH1 (0.41) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL763276 0.92 HRH1 (0.44) KCNH2HRH1CYP2D6CHRM1PROKR1
SCHEMBL763293 0.92 KCNH2 (0.42) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL763530 0.91 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762720 0.90 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762612 0.89 HRH1 (0.46) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL762884 0.89 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL741032 0.88 HRH1 (0.41) KCNH2HRH1CYP2D6CHRM1CYP3A4
SCHEMBL765224 0.88 KCNH2 (0.38) KCNH2HRH1CYP2D6CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed